Molecular Drug Properties

Measurement and Prediction

Chemogenomics in Drug Discovery

A Medicinal Chemistry Perspective

Transporters as Drug Targets

Protein Therapeutics

Animal Models for Human Cancer

Discovery and Development of Novel Therapeutics

Lead Generation

Methods and Strategies

Lead Generation, 2 Volume Set

Methods and Strategies

Fragment-based Drug Discovery

Lessons and Outlook

Thermodynamics and Kinetics of Drug Binding

Predictive Toxicology

From Vision to Reality

In vivo Models for Drug Discovery

Drug Metabolism Prediction

Phosphodiesterases and Their Inhibitors

Natural Products in Medicinal Chemistry

Scaffold Hopping in Medicinal Chemistry

Medicinal Chemistry Approaches to Personalized Medicine

Data Mining in Drug Discovery

Protein-Protein Interactions in Drug Discovery

Protein-Ligand Interactions

Protein Kinases as Drug Targets

Aspartic Acid Proteases as Therapeutic Targets

Antiviral Drug Strategies

Prodrugs and Targeted Delivery

Towards Better ADME Properties

Chemokine Receptors as Drug Targets

Transporters as Drug Carriers

Structure, Function, Substrates

Nuclear Receptors as Drug Targets

Drug Bioavailability

Estimation of Solubility, Permeability, Absorption and Bioavailability

Antitargets

Prediction and Prevention of Drug Side Effects

Mass Spectrometry in Medicinal Chemistry

Applications in Drug Discovery

G Protein-Coupled Receptors as Drug Targets

Analysis of Activation and Constitutive Activity

Ligand Design for G Protein-coupled Receptors

Voltage-Gated Ion Channels as Drug Targets

Protein-Ligand Interactions

From Molecular Recognition to Drug Design

Pharmacophores and Pharmacophore Searches

Chemoinformatics in Drug Discovery

Combinatorial Chemistry

From Theory to Application